Trisubstituted Pyrimidines as Efficacious and Fast-Acting Antimalarials

Author:

Norcross Neil R.1,Baragaña Beatriz1,Wilson Caroline1,Hallyburton Irene1,Osuna-Cabello Maria1,Norval Suzanne1,Riley Jennifer1,Stojanovski Laste1,Simeons Frederick R. C.1,Porzelle Achim1,Grimaldi Raffaella1,Wittlin Sergio23,Duffy Sandra4,Avery Vicky M.4,Meister Stephan5,Sanz Laura6,Jiménez-Díaz Belén6,Angulo-Barturen Iñigo6,Ferrer Santiago6,Martínez María Santos6,Gamo Francisco Javier6,Frearson Julie A.1,Gray David W.1,Fairlamb Alan H.1,Winzeler Elizabeth A.5,Waterson David7,Campbell Simon F.7,Willis Paul7,Read Kevin D.1,Gilbert Ian H.1

Affiliation:

1. Drug Discovery Unit, Division of Biological Chemistry and Drug Discovery, School of Life Sciences, University of Dundee, Dundee, DD1 5EH, U.K.

2. Swiss Tropical and Public Health Institute (Swiss TPH), Socinstrasse 57, 4051 Basel, Switzerland

3. University of Basel, CH-4003 Basel, Switzerland

4. Discovery Biology, Eskitis Institute for Drug Discovery, Griffith University, Nathan, Queensland 4111, Australia

5. Department of Pediatrics, University of California, San Diego School of Medicine, 9500 Gilman Drive, 0741, La Jolla, California 92093, United States

6. Diseases of the Developing World-Tres Cantos Medicines Development Campus, GlaxoSmithKline, c/Severo Ochoa, 2, Tres Cantos, 28760, Madrid, Spain

7. Medicines for Malaria Venture, International Center Cointrin, Entrance G, 3rd Floor, Route de Pré-Bois 20, P.O. Box 1826, CH-1215, Geneva 15, Switzerland

Funder

Wellcome Trust

Medicines for Malaria Venture

MSD Scottish Life Sciences Fund

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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