1. Medicinal Chemistry & Drug Discovery, Department of Pharmacology, University of Oxford, Mansfield Road, Oxford OX1 3QT, U.K.
2. Medicinal
Chemistry, Department of Pharmacy and Pharmacology, University of Bath, Claverton
Down, Bath BA2 7AY, U.K.
3. Laboratory
of Biomolecular Research, Department of Biology and Chemistry, Paul Scherrer Institut, 5232 Villigen PSI, Switzerland
4. Institute
of Metabolism and Systems Research, University of Birmingham, 2nd Floor IBR Tower, Birmingham B15 2TT, U.K.
5. Centre
for Endocrinology, Diabetes and Metabolism, Birmingham Health Partners, Birmingham B15 2TH, U.K.
6. Screening
Technologies Branch, Developmental Therapeutics Program, Division
of Cancer Treatment and Diagnosis, National Cancer Institute, Frederick, Maryland 21702, United States
7. IPSEN, 27 Maple Street, Milford Massachusetts 01757, United States
8. Institut
de Recherche Henri Beaufour, IPSEN, 91966 Les Ulis
Cedex, France
9. University of Basel, Biozentrum, 4056 Basel, Switzerland