A Positive Allosteric Modulator of the Serotonin 5-HT2C Receptor for Obesity-Reference-Cited by-同舟云学术

A Positive Allosteric Modulator of the Serotonin 5-HT2C Receptor for Obesity

Published:2017-11-17 Issue:23 Volume:60 Page:9575-9584
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

García-Cárceles Javier¹^ORCID,Decara Juan M.²,Vázquez-Villa Henar¹^ORCID,Rodríguez Ramón³,Codesido Eva³,Cruces Jacobo³,Brea José⁴,Loza María I.⁴,Alén Francisco²,Botta Joaquin⁵,McCormick Peter J.⁶,Ballesteros Juan A.⁷,Benhamú Bellinda¹^ORCID,Rodríguez de Fonseca Fernando²,López-Rodríguez María L.¹^ORCID

Affiliation:

1. Departamento de Química Orgánica I, Universidad Complutense de Madrid, E-28040 Madrid, Spain

2. Unidad de Gestión Clínica de Salud Mental, Instituto IBIMA, Hospital Regional Universitario, E-29010 Málaga, Spain

3. Galchimia, E-15823 O Pino, A Coruña, Spain

4. Biofarma Research Group, USEF Screening Platform, CIMUS, USC, E-15782 Santiago de Compostela, Spain

5. School of Pharmacy, University of East Anglia, NR4 7TJ Norwich, U.K.

6. School of Veterinary Medicine, University of Surrey, GU2 7XH Guildford, U.K.

7. Vivia Biotech S.L., Parque Científico de Madrid, E-28760 Madrid, Spain

Funder

European Regional Development Fund

Ministerio de Economía y Competitividad

Xunta de Galicia

Comunidad de Madrid

Junta de Andalucía

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b00994

Reference42 articles.

1. Overweight and obesity.Global Health Observatory (GHO) Data;World Health Organization:Geneva, 2017; http://www.who.int/gho/ncd/risk_factors/overweight_text/en/(Sep 25, 2017).

2. Oxidative Stress in Obesity: A Critical Component in Human Diseases

3. Food and Drug Administration's Obesity Drug Guidance Document

4. Past, Present, and Future of Pharmacologic Therapy in Obesity

5. Obesity: Current and potential pharmacotherapeutics and targets

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