Discovery, Structure–Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors-Reference-Cited by-同舟云学术

Discovery, Structure–Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors

Published:2017-08-18 Issue:17 Volume:60 Page:7371-7392
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Joncour Agnès¹,Desroy Nicolas¹^ORCID,Housseman Christopher¹,Bock Xavier¹,Bienvenu Natacha¹,Cherel Laëtitia¹,Labeguere Virginie¹,Peixoto Christophe¹,Annoot Denis¹,Lepissier Luce¹,Heiermann Jörg²,Hengeveld Willem Jan²,Pilzak Gregor²,Monjardet Alain¹,Wakselman Emanuelle¹,Roncoroni Veronique¹,Le Tallec Sandrine¹,Galien René¹,David Christelle¹,Vandervoort Nele³,Christophe Thierry³,Conrath Katja³,Jans Mia³,Wohlkonig Alexandre⁴,Soror Sameh⁴,Steyaert Jan⁴,Touitou Robert¹,Fleury Damien¹,Vercheval Lionel¹,Mollat Patrick¹,Triballeau Nicolas¹,van der Aar Ellen³,Brys Reginald³,Heckmann Bertrand¹

Affiliation:

1. Galapagos SASU, 102 Avenue Gaston Roussel, 93230 Romainville, France

2. Mercachem, Kerkenbos 1013, 6546 Nijmegen, The Netherlands

3. Galapagos NV, Generaal De Wittelaan L11 A3, 2800 Mechelen, Belgium

4. VIB Structural Biology Research Center, Vrije Universiteit Brussel, 1050 Brussel, Belgium

Funder

Agentschap voor Innovatie door Wetenschap en Technologie

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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