Controlling Plasma Stability of Hydroxamic Acids: A MedChem Toolbox-Reference-Cited by-同舟云学术

Controlling Plasma Stability of Hydroxamic Acids: A MedChem Toolbox

Published:2017-10-24 Issue:21 Volume:60 Page:9067-9089
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hermant Paul¹,Bosc Damien¹,Piveteau Catherine¹,Gealageas Ronan¹,Lam BaoVy¹,Ronco Cyril¹,Roignant Matthieu¹,Tolojanahary Hasina¹,Jean Ludovic²,Renard Pierre-Yves²,Lemdani Mohamed³,Bourotte Marilyne¹,Herledan Adrien¹,Bedart Corentin¹,Biela Alexandre¹,Leroux Florence¹,Deprez Benoit¹^ORCID,Deprez-Poulain Rebecca¹⁴^ORCID

Affiliation:

1. Univ. Lille Nord de France, INSERM, Institut Pasteur de Lille, U1177, Drugs and Molecules for Living Systems, F-59000 Lille, France

2. Normandie Université, COBRA, UMR 6014 & FR 3038, Université de Rouen, INSA Rouen, CNRS, F-76821 Mont-Saint-Aignan Cedex, France

3. Univ. Lille, EA 2694, Santé Publique: Épidémiologie et Qualité des Soins, F-59000 Lille, France

4. Institut Universitaire de France, F-75231, Paris, France

Funder

Agence Nationale de la Recherche

Fondation pour la Recherche M??dicale

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b01444

Reference69 articles.

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3. Discovery and Refinement of a New Structural Class of Potent Peptide Deformylase Inhibitors

4. Synthesis/biological evaluation of hydroxamic acids and their prodrugs as inhibitors for Botulinum neurotoxin A light chain

5. Heterocyclic methylsulfone hydroxamic acid LpxC inhibitors as Gram-negative antibacterial agents

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