In Vitro and in Vivo Evaluation of 11C-Labeled Azetidinecarboxylates for Imaging Monoacylglycerol Lipase by PET Imaging Studies

Author:

Cheng Ran12,Mori Wakana3,Ma Longle1ORCID,Alhouayek Mireille4,Hatori Akiko3,Zhang Yiding3,Ogasawara Daisuke5,Yuan Gengyang16,Chen Zhen1,Zhang Xiaofei1,Shi Hang1,Yamasaki Tomoteru3,Xie Lin3,Kumata Katsushi3,Fujinaga Masayuki3,Nagai Yuji7,Minamimoto Takafumi7,Svensson Mona4,Wang Lu1,Du Yunfei2ORCID,Ondrechen Mary Jo6,Vasdev Neil1ORCID,Cravatt Benjamin F.5ORCID,Fowler Christopher4,Zhang Ming-Rong3ORCID,Liang Steven H.1ORCID

Affiliation:

1. Division of Nuclear Medicine and Molecular Imaging, Department of Radiology, Massachusetts General Hospital and Harvard Medical School, Boston, Massachusetts 02114, United States

2. School of Pharmaceutical Science and Technology, Tianjin University, 92 Weijin Road, Nankai District, Tianjin 300072, China

3. Department of Radiopharmaceuticals Development, National Institute of Radiological Sciences, National Institutes for Quantum and Radiological Science and Technology, Chiba 263-8555, Japan

4. Department of Pharmacology and Clinical Neuroscience, Umeå University, SE-901 87 Umeå, Sweden

5. The Skaggs Institute for Chemical Biology and Department of Chemical Physiology, The Scripps Research Institute, SR107 10550 North Torrey Pines Road, La Jolla, California 92037, United States

6. Department of Chemistry and Chemical Biology, Northeastern University, 360 Huntington Avenue, Boston, Massachusetts 02115, United States

7. Department of Functional Brain Imaging Research, National Institute of Radiological Sciences, National Institutes for Quantum and Radiological Science and Technology, Chiba 263-8555, Japan

Funder

Division of Chemistry

Vetenskapsr?det

Division of Molecular and Cellular Biosciences

National Institute on Aging

National Institute on Drug Abuse

China Scholarship Council

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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