Truncated (N)-Methanocarba Nucleosides as Partial Agonists at Mouse and Human A3 Adenosine Receptors: Affinity Enhancement by N6-(2-Phenylethyl) Substitution
Author:
Affiliation:
1. Department of Pharmacology, Medical College of Wisconsin, 8701 Watertown Plank Road, Milwaukee, Wisconsin 53226, United States
2. Institut für Chemie und Biochemie, Freie Universität, Takustraße 3, D-14195 Berlin, Germany
Funder
U.S. Department of Health and Human Services
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c00235
Reference69 articles.
1. A3Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy
2. The A3Adenosine Receptor: History and Perspectives
3. Agonists and Antagonists: Molecular Mechanisms and Therapeutic Applications
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