First Potent Macrocyclic A<sub>3</sub> Adenosine Receptor Agonists Reveal G-Protein and β-Arrestin2 Signaling Preferences-Reference-Cited by-同舟云学术

First Potent Macrocyclic A₃ Adenosine Receptor Agonists Reveal G-Protein and β-Arrestin2 Signaling Preferences

Published:2023-08-08 Issue:9 Volume:6 Page:1288-1305
ISSN:2575-9108
Container-title:ACS Pharmacology & Translational Science
language:en
Short-container-title:ACS Pharmacol. Transl. Sci.

Author:

Tosh Dilip K.¹,Fisher Courtney L.²,Salmaso Veronica¹³,Wan Tina C.²,Campbell Ryan G.¹,Chen Eric¹,Gao Zhan-Guo¹,Auchampach John A.²^ORCID,Jacobson Kenneth A.¹^ORCID

Affiliation:

1. Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Disease, National Institutes of Health, 9000 Rockville Pike, Bethesda, Maryland 20892, United States

2. Department of Pharmacology & Toxicology and the Cardiovascular Center, Medical College of Wisconsin, 8701 Watertown Plank Road, Milwaukee, Wisconsin 53226, United States

3. Molecular Modeling Section, Department of Pharmaceutical and Pharmacological Sciences, University of Padua, Padua 35131, Italy

Funder

National Institute of Diabetes and Digestive and Kidney Diseases

National Heart, Lung, and Blood Institute

Publisher

American Chemical Society (ACS)

Subject

Pharmacology (medical),Pharmacology

Link

https://pubs.acs.org/doi/pdf/10.1021/acsptsci.3c00126

Reference79 articles.

1. A3Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy

2. Adenosine Metabotropic Receptors in Chronic Pain Management

3. Namodenoson in Advanced Hepatocellular Carcinoma and Child–Pugh B Cirrhosis: Randomized Placebo-Controlled Clinical Trial

4. A3 Adenosine Receptor Agonist Reduces Brain Ischemic Injury and Inhibits Inflammatory Cell Migration in Rats

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