Assay-Dependent Inverse Agonism at the A<sub>3</sub> Adenosine Receptor: When Neutral Is Not Neutral-Reference-Cited by-同舟云学术

Assay-Dependent Inverse Agonism at the A₃ Adenosine Receptor: When Neutral Is Not Neutral

Published:2023-08-09 Issue:9 Volume:6 Page:1266-1274
ISSN:2575-9108
Container-title:ACS Pharmacology & Translational Science
language:en
Short-container-title:ACS Pharmacol. Transl. Sci.

Author:

Pottie Eline¹,Suresh R. Rama²^ORCID,Jacobson Kenneth A.²^ORCID,Stove Christophe P.¹^ORCID

Affiliation:

1. Laboratory of Toxicology, Department of Bioanalysis, Faculty of Pharmaceutical Sciences, Ghent University, Campus Heymans, Ottergemsesteenweg 460, B-9000 Ghent, Belgium

2. Laboratory of Bioorganic Chemistry, National Institute of Diabetes & Digestive & Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20802, United States

Funder

National Institute of Diabetes and Digestive and Kidney Diseases

Publisher

American Chemical Society (ACS)

Subject

Pharmacology (medical),Pharmacology

Link

https://pubs.acs.org/doi/pdf/10.1021/acsptsci.3c00071

Reference41 articles.

1. A3Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy

2. Molecular dissection of the human A 3 adenosine receptor coupling with β-arrestin2

3. The A3Adenosine Receptor: History and Perspectives

4. Biased agonism at adenosine receptors

5. Nucleotide P2Y1 receptor agonists are in vitro and in vivo prodrugs of A1/A3 adenosine receptor agonists: implications for roles of P2Y1 and A1/A3 receptors in physiology and pathology

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