Structural Characterization of Agonist Binding to an A3 Adenosine Receptor through Biomolecular Simulations and Mutagenesis Experiments-Reference-Cited by-同舟云学术

Structural Characterization of Agonist Binding to an A3 Adenosine Receptor through Biomolecular Simulations and Mutagenesis Experiments

Published:2019-09-10 Issue:19 Volume:62 Page:8831-8846
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Stamatis Dimitrios¹,Lagarias Panagiotis¹,Barkan Kerry²,Vrontaki Eleni¹,Ladds Graham²,Kolocouris Antonios¹^ORCID

Affiliation:

1. Division of Pharmaceutical Chemistry, Department of Pharmacy, School of Health Sciences, National and Kapodistrian University of Athens, Panepistimiopolis-Zografou, 15771 Athens, Greece

2. Department of Pharmacology, University of Cambridge, Tennis Court Road, CB2 1PD Cambridge U.K.

Funder

State Scholarships Foundation

Leverhulme Trust

Biotechnology and Biological Sciences Research Council

Chiesi Hellas

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.9b01164

Reference93 articles.

1. International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and Classification of Adenosine Receptors—An Update

2. Adenosine receptors: targets for future drugs

3. Adenosine as an Antiarrhythmic Agent

4. Adenosine receptors as drug targets — what are the challenges?

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