Protein Stability Effects in Aggregate-Based Enzyme Inhibition
Author:
Affiliation:
1. Department of Pharmaceutical Chemistry, University of California, San Francisco, 1700 Fourth Street, San Francisco, California 94143-2550, United States
Funder
National Institute of General Medical Sciences
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.9b01019
Reference36 articles.
1. A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening
2. Identification and Prediction of Promiscuous Aggregating Inhibitors among Known Drugs
3. Concentration and pH Dependent Aggregation of Hydrophobic Drug Molecules and Relevance to Oral Bioavailability
4. Mechanisms of Specific versus Nonspecific Interactions of Aggregation-Prone Inhibitors and Attenuators
5. Internal Structure and Preferential Protein Binding of Colloidal Aggregates
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