Synthesis, Biological Properties, and Molecular Modeling Investigation of the First Potent, Selective, and Water-Soluble Human A3 Adenosine Receptor Antagonist-Reference-Cited by-同舟云学术

Synthesis, Biological Properties, and Molecular Modeling Investigation of the First Potent, Selective, and Water-Soluble Human A3 Adenosine Receptor Antagonist

Published:2002-07-16 Issue:17 Volume:45 Page:3579-3582
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Maconi Anna¹,Pastorin Giorgia¹,Da Ros Tatiana¹,Spalluto Giampiero¹,Gao Zhan-guo¹,Jacobson Kenneth A.¹,Baraldi Pier Giovanni¹,Cacciari Barbara¹,Varani Katia¹,Moro Stefano¹,Borea Pier Andrea¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche, Università degli Studi di Trieste, Piazzale Europa 1, I-34127 Trieste, Italy, Molecular Recognition Section, LBC, National Institute of Diabetes & Digestive & Kidney Diseases, National Institutes of Health, Building 8A, Room B1A-19, Bethesda, Maryland 20892-0810, Dipartimento di Scienze Farmaceutiche, Università degli Studi di Ferrara, Via Fossato di Mortara 17-19, I-44100 Ferrara, Italy, Dipartimento di Medicina Clinica e Sperimentale-Sezione di Farmacologia,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm020974x

Reference27 articles.

1. Molecular cloning and characterization of the human A3 adenosine receptor.

2. Recent developments in selective agonists and antagonists acting at purine and pyrimidine receptors

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