Meta-Substituted Aryl(thio)ethers as Potent Partial Agonists (or Antagonists) for the Histamine H3 Receptor Lacking a Nitrogen Atom in the Side Chain-Reference-Cited by-同舟云学术

Meta-Substituted Aryl(thio)ethers as Potent Partial Agonists (or Antagonists) for the Histamine H3 Receptor Lacking a Nitrogen Atom in the Side Chain

Published:2004-05-08 Issue:12 Volume:47 Page:3264-3274
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Pelloux-Léon Nadia¹,Fkyerat Abdellatif¹,Piripitsi Antonia¹,Tertiuk Wasyl¹,Schunack Walter¹,Stark Holger¹,Garbarg Monique¹,Ligneau Xavier¹,Arrang Jean-Michel¹,Schwartz Jean-Charles¹,Ganellin C. Robin¹

Affiliation:

1. Department of Chemistry, University College London, 20 Gordon Street, London WC1H 0AJ, England, Institut für Pharmazie, Freie Universität Berlin, Königin-Luise-Strasse 2 + 4, 14195 Berlin (Dahlem), Germany, Biozentrum, Institut für Pharmazeutische Chemie, Johann Wolfgang Goethe-Universität, Marie-Curie-Strasse 9, 60439 Frankfurt/M, Germany, Laboratoire Bioprojet, 30 Rue des Francs-Bourgeois, 75003 Paris, France, and Unité 109 de Neurobiologie et Pharmacologie Moléculaire, Centre Paul Broca de l'INSERM,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm031141p

Reference71 articles.

1. Three loci related to the src oncogene and tyrosine-specific protein kinase activity in Drosophila

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3. Modulation of neurotransmitter releaseviahistamine H3heteroreceptors

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