Investigation of the Histamine H3 Receptor Binding Site. Design and Synthesis of Hybrid Agonists with a Lipophilic Side Chain
Author:
Affiliation:
1. Pharmaceutical Research Center, Meiji Seika Kaisha, Ltd., 760 Morooka-cho, Kohoku-ku, Yokohama 222-8567, Japan
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm100643t
Reference39 articles.
1. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor
2. Autoregulation of histamine release in brain by presynaptic H3-receptors
3. Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors
4. Possible participation of histamine H3 receptors in the modulation of noradrenaline release from rat spinal cord slices
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