4-Aminoquinolone Piperidine Amides: Noncovalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial Activity
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Published:2014-06-11
Issue:12
Volume:57
Page:5419-5434
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ISSN:0022-2623
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Container-title:Journal of Medicinal Chemistry
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language:en
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Short-container-title:J. Med. Chem.
Author:
Naik Maruti, Humnabadkar Vaishali, Tantry Subramanyam J., Panda Manoranjan, Narayan Ashwini, Guptha Supreeth, Panduga Vijender, Manjrekar Praveena, Jena Lalit kumar, Koushik Krishna, Shanbhag Gajanan, Jatheendranath Sandesh, Manjunatha M. R., Gorai Gopinath, Bathula Chandramohan, Rudrapatna Suresh, Achar Vijayashree, Sharma Sreevalli, Ambady Anisha, Hegde Naina, Mahadevaswamy Jyothi, Kaur Parvinder, Sambandamurthy Vasan K., Awasthy Disha, Narayan Chandan, Ravishankar Sudha, Madhavapeddi Prashanti, Reddy Jitendar, Prabhakar KR, Saralaya Ramanatha, Chatterji Monalisa, Whiteaker James, McLaughlin Bob, Chiarelli Laurent R.1, Riccardi Giovanna1, Pasca Maria Rosalia1, Binda Claudia1, Neres João2, Dhar Neeraj2, Signorino-Gelo François2, McKinney John D.2, Ramachandran Vasanthi, Shandil Radha, Tommasi Ruben, Iyer Pravin S., Narayanan Shridhar, Hosagrahara Vinayak, Kavanagh Stefan3, Dinesh Neela, Ghorpade Sandeep R.
Affiliation:
1. Department
of Biology and Biotechnology “Lazzaro Spallanzani”, University of Pavia, 27100 Pavia, Italy 2. École Polytechnique Fédérale de Lausanne, 1015 Lausanne, Switzerland 3. Safety Assessment, AstraZeneca, Alderley
Park, Macclesfield, Cheshire SK10 2NA, United Kingdom
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Cited by
80 articles.
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