Discovery of 1,2,3-triazole incorporated indole-piperazines as potent antitubercular agents: Design, synthesis, in vitro biological evaluation, molecular docking and ADME studies-Reference-Cited by-同舟云学术

Discovery of 1,2,3-triazole incorporated indole-piperazines as potent antitubercular agents: Design, synthesis, in vitro biological evaluation, molecular docking and ADME studies

Published:2024-01 Issue: Volume:98 Page:117562
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Reddyrajula Rajkumar,Etikyala Umadevi,Manga Vijjulatha,kumar Dalimba Udaya

Funder

National Institute of Technology Karnataka, Surathkal

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference54 articles.

1. Functional genetic diversity among Mycobacterium tuberculosis complex clinical isolates: delineation of conserved core and lineage-specific transcriptomes during intracellular survival;Homolka;PLoS Pathog,2010

2. Synthesis and pharmacokinetic evaluation of siderophore biosynthesis inhibitors for Mycobacterium tuberculosis;Nelson;J Med Chem,2015

3. WHO’s global tuberculosis report 2022;Bagcchi;The Lancet Microbe,2023

4. Synthetic account of indoles in search of potential anti-mycobacterial agents: a review and future insights;Bhakhar;J Mol Struct,2022

5. Indole chalcones: Design, synthesis, in vitro and in silico evaluation against Mycobacterium tuberculosis;Ramesh;Eur J Med Chem,2020

Cited by 4 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. N-Acyl phenothiazines as mycobacterial ATP synthase inhibitors: Rational design, synthesis and in vitro evaluation against drug sensitive, RR and MDR-TB;Bioorganic Chemistry;2024-10

2. Design, synthesis and molecular docking of 5-fluoro indole derivatives as inhibitors of PI3K/Akt signalling pathway in cervical cancer;Journal of Molecular Structure;2024-09

3. Antitüberküler Bileşiklerde Piperazin Yapısı;Hacettepe University Journal of the Faculty of Pharmacy;2024-09-01

4. Design, Synthesis and In vitro Antitubercular Effect of New Chalcone Derivatives Coupled with 1,2,3‐Triazoles: A Computational Docking Techniques;Chemistry & Biodiversity;2024-04-02