Trastuzumab Labeled to High Specific Activity with 111In by Site-Specific Conjugation to a Metal-Chelating Polymer Exhibits Amplified Auger Electron-Mediated Cytotoxicity on HER2-Positive Breast Cancer Cells

Author:

Ngo Ndjock Mbong Ghislaine1,Lu Yijie2,Chan Conrad1,Cai Zhongli1,Liu Peng2,Boyle Amanda J.1,Winnik Mitchell A.2,Reilly Raymond M.134

Affiliation:

1. Department of Pharmaceutical Sciences, University of Toronto, 144 College Street, Toronto, ON M5S 3M2, Canada

2. Department of Chemistry, University of Toronto, 80 St. George Street, Toronto, ON M5S 3H6, Canada

3. Department of Medical Imaging, University of Toronto, 263 McCaul Street, Toronto, ON M5T 1W7, Canada

4. Toronto General Research Institute, University Health Network, 200 Elizabeth Street, Toronto, ON M5G 2C4, Canada

Funder

Canadian Institutes of Health Research

Canadian Breast Cancer Research Alliance

Canadian Cancer Society

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

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