A Scalable Route to the SMO Receptor Antagonist SEN826: Benzimidazole Synthesis via Enhanced in Situ Formation of the Bisulfite–Aldehyde Complex
Author:
Affiliation:
1. Process Chemistry Unit, Siena Biotech SpA, 53100 Siena, Italy
2. Compound Management & Analysis Unit, Siena Biotech SpA, 53100 Siena, Italy
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/op4002092
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