Practical Asymmetric Synthesis of a Calcitonin Gene-Related Peptide (CGRP) Receptor Antagonist Ubrogepant-Reference-Cited by-同舟云学术

Practical Asymmetric Synthesis of a Calcitonin Gene-Related Peptide (CGRP) Receptor Antagonist Ubrogepant

Published:2017-11-02 Issue:11 Volume:21 Page:1851-1858
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Yasuda Nobuyoshi¹^ORCID,Cleator Ed²,Kosjek Birgit¹,Yin Jianguo¹,Xiang Bangping¹,Chen Frank¹,Kuo Shen-Chun¹,Belyk Kevin¹,Mullens Peter R.²,Goodyear Adrian²,Edwards John S.²,Bishop Brian²,Ceglia Scott³,Belardi Justin³,Tan Lushi¹,Song Zhiguo J.¹,DiMichele Lisa¹,Reamer Robert¹,Cabirol Fabien L.⁴,Tang Weng Lin⁴,Liu Guiquan⁵

Affiliation:

1. Department of Process Chemistry, MRL, 126 East Lincoln Avenues, Rahway, New Jersey 07065, United States

2. Department of Process Chemistry, MSD Research Laboratories, Hertford Road, Hoddesdon, Hertford, Hertfordshire EN11 9BU, United Kingdom

3. Department of Process Chemistry, MRL, 770 Sumneytown Pike, West Point, Pennsylvania 19486, United States

4. Codexis, Inc., 200 Penobscot Drive, Redwood City, California 94063, United States

5. Shanghai SynTheAll Pharmaceutical Co. Ltd., 9 Yuegong Road, Jinshan District, Shanghai, 201507, China

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.7b00293

Reference20 articles.

1. Migraine — Current Understanding and Treatment

2. The Global Burden of Headache: A Documentation of Headache Prevalence and Disability Worldwide

3. Cardiovascular Safety of 5Ht1B/1D Agonists—Is There a Cause for Concern?

4. Targeting a family B GPCR/RAMP receptor complex: CGRP receptor antagonists and migraine

5. Calcitonin Gene-Related Peptide Receptor Antagonists: New Therapeutic Agents for Migraine

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