Amination of a Green Solvent via Immobilized Biocatalysis for the Synthesis of Nemtabrutinib

Author:

Prier Christopher K.1,Camacho Soto Karla1,Forstater Jacob H.1,Kuhl Nadine1ORCID,Kuethe Jeffrey T.1,Cheung-Lee Wai Ling1ORCID,Di Maso Michael J.1ORCID,Eberle Claire M.1,Grosser Shane T.1,Ho Hsing-I1,Hoyt Erik2,Maguire Anne1ORCID,Maloney Kevin M.1ORCID,Makarewicz Amanda1,McMullen Jonathan P.1ORCID,Moore Jeffrey C.1ORCID,Murphy Grant S.1,Narsimhan Karthik1,Pan Weilan1,Rivera Nelo R.2ORCID,Saha-Shah Anumita2ORCID,Thaisrivongs David A.1ORCID,Verma Deeptak3ORCID,Wyatt Adeya1,Zewge Daniel2ORCID

Affiliation:

1. Process Research and Development, Merck & Co., Inc., Rahway, New Jersey 07065, United States

2. Analytical Research and Development, Merck & Co., Inc., Rahway, New Jersey 07065, United States

3. Computational and Structural Chemistry, Merck & Co., Inc., Rahway, New Jersey 07065, United States

Funder

Merck Sharp and Dohme

Publisher

American Chemical Society (ACS)

Subject

Catalysis,General Chemistry

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