Discovery of β2 Adrenergic Receptor Ligands Using Biosensor Fragment Screening of Tagged Wild-Type Receptor

Author:

Aristotelous Tonia1,Ahn Seungkirl2,Shukla Arun K.2,Gawron Sylwia1,Sassano Maria F.3,Kahsai Alem W.2,Wingler Laura M.2,Zhu Xiao2,Tripathi-Shukla Prachi2,Huang Xi-Ping3,Riley Jennifer1,Besnard Jérémy1,Read Kevin D.1,Roth Bryan L.34,Gilbert Ian H.1,Hopkins Andrew L.1,Lefkowitz Robert J.256,Navratilova Iva1

Affiliation:

1. Division of Biological Chemistry and Drug Discovery, College of Life Sciences, University of Dundee, Dow Street, Dundee DD1 5EH, United Kingdom

2. Department of Medicine, Duke University Medical Center, Durham, North Carolina 27710, United States

3. NIMH Psychoactive Drug Screening Program, Department of Pharmacology, The University of North Carolina Chapel Hill School of Medicine, Chapel Hill, North Carolina 27759, United States

4. Department of Pharmacology and Division of Chemical Biology and Medicinal Chemistry, The University of North Carolina Chapel Hill School of Medicine, Chapel Hill, North Carolina 27759, United States

5. Howard Hughes Medical Institute, Duke University Medical Center, Durham, North Carolina 27710, United States

6. Department of Biochemistry, Duke University Medical Center, Durham, North Carolina 27710, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

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