Fragment Screening at Adenosine-A3 Receptors in Living Cells Using a Fluorescence-Based Binding Assay-Reference-Cited by-同舟云学术

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Fragment Screening at Adenosine-A3 Receptors in Living Cells Using a Fluorescence-Based Binding Assay

Published:2012-09 Issue:9 Volume:19 Page:1105-1115
ISSN:1074-5521
Container-title:Chemistry & Biology
language:en
Short-container-title:Chemistry & Biology

Author:

Stoddart Leigh A.,Vernall Andrea J.,Denman Jessica L.,Briddon Stephen J.,Kellam Barrie,Hill Stephen J.

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,Molecular Medicine,General Medicine,Biochemistry

Reference42 articles.

1. β-arrestin-mediated activation of MAPK by inverse agonists reveals distinct active conformations for G protein-coupled receptors;Azzi;Proc. Natl. Acad. Sci. USA,2003

2. Multiple GPCR conformations and signalling pathways: implications for antagonist affinity estimates;Baker;Trends Pharmacol. Sci.,2007

3. Pharmacological characterization of CGP 12177 at the human β(2)-adrenoceptor;Baker;Br. J. Pharmacol.,2002

4. Agonist and inverse agonist actions of β-blockers at the human β2-adrenoceptor provide evidence for agonist-directed signalling;Baker;Mol. Pharm.,2003

5. The fragment-approach: an update;Bartoli;Drug Discov. Today. Technol.,2006

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