An Efficient Process of Racemization of 3-(Carbamoylmethyl)-5-methylhexanoic acid: A Pregabalin Intermediate
Author:
Affiliation:
1. Emcure Pharmaceuticals Ltd, R & D Centre, Plot No.12/2, F-II Block, M.I.D.C., Pimpri, Pune - 411018, India
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/op900064x
Reference10 articles.
1. Structure−Activity Relationships of Pregabalin and Analogues That Target the α2-δ Protein
2. Chemical Development of CI-1008, an Enantiomerically Pure Anticonvulsant
3. Huckabee, B.; Keith, S.; Denis, M.World Patent, WO96/38405, 1996.
4. Stereoselective synthesis of γ-amino acids
5. Development of a Chemoenzymatic Manufacturing Process for Pregabalin
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