Structure−Activity Relationships of Pregabalin and Analogues That Target the α2-δ Protein-Reference-Cited by-同舟云学术

Structure−Activity Relationships of Pregabalin and Analogues That Target the α2-δ Protein

Published:2005-02-17 Issue:7 Volume:48 Page:2294-2307
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Belliotti Thomas R.¹,Capiris Thomas¹,Ekhato I. Victor¹,Kinsora Jack J.¹,Field Mark J.¹,Heffner Thomas G.¹,Meltzer Leonard T.¹,Schwarz Jacob B.¹,Taylor Charles P.¹,Thorpe Andrew J.¹,Vartanian Mark G.¹,Wise Lawrence D.¹,Zhi-Su Ti¹,Weber Mark L.¹,Wustrow David J.¹

Affiliation:

1. Pfizer Global Research and Development, Michigan Laboratories, Ann Arbor Campus, Ann Arbor, MI, 48105, Sandwich Laboratories, Sandwich, Kent CT13 9NJ UK, Nagoya Laboratories, 5-2 Takatoy-Cho, Chita-gun Aichi, 470-2393 Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049762l

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4. 3-Alkyl-4-aminobutyric acids: the first class of anticonvulsant agents that activates L-glutamic acid decarboxylase

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