Optimization of Substituted N-3-Benzylimidazoquinazolinone Sulfonamides as Potent and Selective PDE5 Inhibitors-Reference-Cited by-同舟云学术

Optimization of Substituted N-3-Benzylimidazoquinazolinone Sulfonamides as Potent and Selective PDE5 Inhibitors

Published:2000-11-22 Issue:26 Volume:43 Page:5037-5043
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Rotella David P.¹,Sun Zhong¹,Zhu Yeheng¹,Krupinski John¹,Pongrac Ronald¹,Seliger Laurie¹,Normandin Diane¹,Macor John E.¹

Affiliation:

1. Departments of Discovery Chemistry and Metabolic and Cardiovascular Drug Discovery, Bristol-Myers Squibb Pharmaceutical Research Institute, P.O. Box 5400, Princeton, New Jersey 08543-5400

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm000336j

Reference14 articles.

1. Impotence and Its Medical and Psychosocial Correlates: Results of the Massachusetts Male Aging Study

2. 4-(3-Chloro-4-methoxybenzyl)aminophthalazines: Synthesis and Inhibitory Activity toward Phosphodiesterase 5

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