Route Design and Development of a MET Kinase Inhibitor: A Copper-Catalyzed Preparation of an N1-Methylindazole-Reference-Cited by-同舟云学术

Route Design and Development of a MET Kinase Inhibitor: A Copper-Catalyzed Preparation of an N1-Methylindazole

Published:2014-03-18 Issue:4 Volume:18 Page:501-510
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Kallman Neil J.¹,Liu Chin¹,Yates Matthew H.¹,Linder Ryan J.¹,Ruble J. Craig¹,Kogut Eugene F.¹,Patterson Lawrence E.¹,Laird Dana L. T.¹,Hansen Marvin M.¹

Affiliation:

1. Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, Indiana 46285, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op400317z

Reference28 articles.

1. Process Development and Large-Scale Synthesis of a c-Met Kinase Inhibitor

2. Development of c-MET pathway inhibitors

3. LY2801653 is an orally bioavailable multi-kinase inhibitor with potent activity against MET, MST1R, and other oncoproteins, and displays anti-tumor activities in mouse xenograft models

4. Über Bildung von Indazolkörpern aus orthomethylierten Anilinbasen

5. Aromatische Diazoniumsalze, VIII: Der Mechanismus der Indazolsynthese aus o ‐Toluoldiazoniumsalzen

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