Process Development for a 1<i>H</i>-Indazole Synthesis Using an Intramolecular Ullmann-Type Reaction-Reference-Cited by-同舟云学术

Process Development for a 1H-Indazole Synthesis Using an Intramolecular Ullmann-Type Reaction

Published:2023-03-23 Issue:7 Volume:88 Page:4209-4223
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Day Jon I.¹^ORCID,Allen-Moyer Katherine N.²,Cole Kevin P.¹^ORCID

Affiliation:

1. Synthetic Molecule Design and Development, Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana 46285, United States

2. Statistics − Discovery/Development, Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN, 46285. Current: Social and Scientific Systems, Inc., A DLH Holdings Corp. Company, Durham, North Carolina 27703, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.2c02771

Reference60 articles.

1. Über Bildung von Indazolkörpern aus orthomethylierten Anilinbasen

2. Ren, Z. S.; Zhou, J.; Xu, Q. Tetrahydropyrazolo-pyridinyl-dihydrolmidazolone or Tetrahydropyrazolo-pyridinyl-dihydrolmidazolone Compounds and Methods of Using Same. WO 2022/017338 Al, 2022.

3. Route Design and Development of a MET Kinase Inhibitor: A Copper-Catalyzed Preparation of an N1-Methylindazole

4. Directed Ortho Metalation in 2021: A Tribute to Victor Snieckus (August 1, 1937–December 18, 2020)

Cited by 2 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Construction of C–X (X = N, O) bonds from benzyl alcohols via Cu-BTC-catalyzed oxidative coupling;Catalysis Science & Technology;2024

2. Cu-Mediated Cyclization to Form 1H-Indazoles;Synfacts;2023-09-14