Discovery of Novel P1 Groups for Coagulation Factor VIIa Inhibition Using Fragment-Based Screening-Reference-Cited by-同舟云学术

Discovery of Novel P1 Groups for Coagulation Factor VIIa Inhibition Using Fragment-Based Screening

Published:2015-03-12 Issue:6 Volume:58 Page:2799-2808
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Cheney Daniel L.¹,Bozarth Jeffrey M.¹,Metzler William J.²,Morin Paul E.²,Mueller Luciano²,Newitt John A.²,Nirschl Alexandra H.¹,Rendina Alan R.¹,Tamura James K.²,Wei Anzhi¹,Wen Xiao¹,Wurtz Nicholas R.¹,Seiffert Dietmar A.¹,Wexler Ruth R.¹,Priestley E. Scott¹

Affiliation:

1. Bristol-Myers Squibb Co., Research and Development, 311 Pennington-Rocky Hill Road, Pennington, New Jersey 08543, United States

2. Bristol-Myers Squibb, Research & Development, P.O. Box 4000, Princeton, New Jersey 08543-4000, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm501982k

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