Extending the Detection Limit in Fragment Screening of Proteins Using Reverse Micelle Encapsulation-Reference-Cited by-同舟云学术

Extending the Detection Limit in Fragment Screening of Proteins Using Reverse Micelle Encapsulation

Published:2019-10-03 Issue: Volume: Page:
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Fuglestad Brian¹,Kerstetter Nicole E.²^ORCID,Bédard Sabrina¹,Wand A. Joshua¹²^ORCID

Affiliation:

1. Johnson Research Foundation and Department of Biochemistry and Biophysics, University of Pennsylvania, Perelman School of Medicine, Philadelphia, Pennsylvania 19104, United States

2. Graduate Group in Biochemistry and Molecular Biophysics, University of Pennsylvania, Philadelphia, Pennsylvania 19104, United States

Funder

National Cancer Institute

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acschembio.9b00537

Reference56 articles.

1. Twenty years on: the impact of fragments on drug discovery

2. A ‘Rule of Three’ for fragment-based lead discovery?

3. Reaching for high-hanging fruit in drug discovery at protein–protein interfaces

4. The maximal affinity of ligands

5. On the attribution and additivity of binding energies

Cited by 8 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Ligandability at the Membrane Interface of GPx4 Revealed through a Reverse Micelle Fragment Screening Platform;JACS Au;2024-06-26

2. An NMR Approach for Investigating Membrane Protein–Lipid Interactions Using Native Reverse Micelles;BIO-PROTOCOL;2024

3. Investigating protein‐membrane interactions using native reverse micelles constructed from naturally sourced lipids;Protein Science;2023-10-16

4. Membrane-Mimicking Reverse Micelles for High-Resolution Interfacial Study of Proteins and Membranes;Langmuir;2022-03-17

5. Small Glycols Discover Cryptic Pockets on Proteins for Fragment-Based Approaches;Journal of Chemical Information and Modeling;2021-02-11