Design, Synthesis, and Biological Evaluation of a Series of Benzo[de][1,7]naphthyridin-7(8H)-ones Bearing a Functionalized Longer Chain Appendage as Novel PARP1 Inhibitors-Reference-Cited by-同舟云学术

Design, Synthesis, and Biological Evaluation of a Series of Benzo[de][1,7]naphthyridin-7(8H)-ones Bearing a Functionalized Longer Chain Appendage as Novel PARP1 Inhibitors

Published:2013-03-21 Issue:7 Volume:56 Page:2885-2903
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ye Na¹,Chen Chuan-Huizi¹,Chen TianTian¹,Song Zilan¹,He Jin-Xue¹,Huan Xia-Juan¹,Song Shan-Shan¹,Liu Qiufeng¹,Chen Yi¹,Ding Jian¹,Xu Yechun¹,Miao Ze-Hong¹,Zhang Ao¹

Affiliation:

1. CAS Key Laboratory of Receptor Research, and Synthetic Organic & Medicinal Chemistry Laboratory, ‡State Key Laboratory of Drug Research, and §CAS Key Laboratory of Receptor Research, and Drug Discovery and Design Center, Shanghai Institute of Materia Medica (SIMM), Chinese Academy of Sciences, Shanghai, China 201203

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm301825t

Reference64 articles.

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4. Poly(ADP-ribose): novel functions for an old molecule

5. Toward specific functions of poly(ADP-ribose) polymerase-2

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