Optimized Chemical Probes for REV-ERBα-Reference-Cited by-同舟云学术

Optimized Chemical Probes for REV-ERBα

Published:2013-05-23 Issue:11 Volume:56 Page:4729-4737
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Trump Ryan P.¹,Bresciani Stefano²,Cooper Anthony W. J.³,Tellam James P.²,Wojno Justyna²,Blaikley John⁴,Orband-Miller Lisa A.¹,Kashatus Jennifer A.¹,Boudjelal Mohamed³,Dawson Helen C.¹,Loudon Andrew⁵,Ray David⁴,Grant Daniel¹,Farrow Stuart N.³,Willson Timothy M.¹,Tomkinson Nicholas C. O.²

Affiliation:

1. Molecular Discovery Research, GlaxoSmithKline, Research Triangle Park, North Carolina 27709-3398, United States

2. WestCHEM, Department of Pure and Applied Chemistry, Thomas Graham Building, University of Strathclyde, Glasgow, G1 1XL, U.K.

3. Molecular Discovery Research, GlaxoSmithKline, Medicines Research Centre, Hertfordshire, SG1 2NY, U.K.

4. Faculty of Medical and Human Sciences, University of Manchester, Manchester, M13 9PT, U.K.

5. Faculty of Life Sciences, University of Manchester, Manchester, M13 9PT, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm400458q

Reference18 articles.

1. GSK4112, a Small Molecule Chemical Probe for the Cell Biology of the Nuclear Heme Receptor Rev-erbα

2. Circadian Integration of Metabolism and Energetics

3. The genetics of mammalian circadian order and disorder: implications for physiology and disease

4. Suprachiasmatic Nucleus: Cell Autonomy and Network Properties

5. Transcriptional coactivator PGC-1α integrates the mammalian clock and energy metabolism

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