GSK4112, a Small Molecule Chemical Probe for the Cell Biology of the Nuclear Heme Receptor Rev-erbα-Reference-Cited by-同舟云学术

GSK4112, a Small Molecule Chemical Probe for the Cell Biology of the Nuclear Heme Receptor Rev-erbα

Published:2010-08-13 Issue:10 Volume:5 Page:925-932
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Grant Daniel¹,Yin Lei²,Collins Jon L.¹,Parks Derek J.¹,Orband-Miller Lisa A.¹,Wisely G. Bruce¹,Joshi Shree²,Lazar Mitchell A.²,Willson Timothy M.¹,Zuercher William J.¹

Affiliation:

1. GlaxoSmithKline, Research Triangle Park, North Carolina, 27707

2. Division of Endocrinology, Diabetes, and Metabolism, Department of Medicine and Department of Genetics, and The Institute for Diabetes, Obesity, and Metabolism, University of Pennsylvania School of Medicine, Philadelphia, Pennsylvania 19104

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/cb100141y

Reference28 articles.

1. Transcriptional coactivator PGC-1α integrates the mammalian clock and energy metabolism

2. Identification of heme as the ligand for the orphan nuclear receptors REV-ERBα and REV-ERBβ

3. Structural Insight into the Constitutive Repression Function of the Nuclear Receptor Rev-erbβ

4. Rev-erbα, a Heme Sensor That Coordinates Metabolic and Circadian Pathways

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