Probing Structural Requirements of Positive Allosteric Modulators of the M4 Muscarinic Receptor-Reference-Cited by-同舟云学术

Probing Structural Requirements of Positive Allosteric Modulators of the M4 Muscarinic Receptor

Published:2013-10-11 Issue:20 Volume:56 Page:8196-8200
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Huynh Tracey¹,Valant Celine¹,Crosby Ian T.¹,Sexton Patrick M.¹,Christopoulos Arthur¹,Capuano Ben¹

Affiliation:

1. Medicinal Chemistry and ‡Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381-399 Royal Parade, Parkville VIC 3052, Australia

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm401032k

Reference17 articles.

1. Immunological localization of m1–m5 muscarinic acetylcholine receptors in peripheral tissues and brain

2. Selective Muscarinic Receptor Agonist Xanomeline as a Novel Treatment Approach for Schizophrenia

3. Allosteric binding sites on muscarinic receptors

4. Allosteric Modulation of Seven Transmembrane Spanning Receptors: Theory, Practice, and Opportunities for Central Nervous System Drug Discovery

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