Synthesis and Preliminary Evaluation of 11 C‐Labeled VU0467485/AZ13713945 and Its Analogues for Imaging Muscarinic Acetylcholine Receptor Subtype 4-Reference-Cited by-同舟云学术

Synthesis and Preliminary Evaluation of 11 C‐Labeled VU0467485/AZ13713945 and Its Analogues for Imaging Muscarinic Acetylcholine Receptor Subtype 4

Published:2018-12-27 Issue:3 Volume:14 Page:303-309
ISSN:1860-7179
Container-title:ChemMedChem
language:en
Short-container-title:ChemMedChem

Author:

Deng Xiaoyun¹,Hatori Akiko²,Chen Zhen¹,Kumata Katsushi²,Shao Tuo¹,Zhang Xiaofei¹,Yamasaki Tomoteru²,Hu Kuan²,Yu Qingzhen¹,Ma Longle¹,Wang Gangqiang³,Wang Lu¹⁴,Shao Yihan⁵,Josephson Lee¹,Sun Shaofa³,Zhang Ming‐Rong²,Liang Steven¹^ORCID

Affiliation:

1. Department of Radiology, Division of Nuclear Medicine and Molecular ImagingMassachusetts General Hospital and Harvard Medical School 55 Fruit Street Boston MA 02114 USA

2. Department of Radiopharmaceuticals Development, National Institute of Radiological SciencesNational Institutes for Quantum and Radiological Science and Technology Chiba 263-8555 Japan

3. Hubei Collaborative Innovation Centre for Non-power Nuclear Technology, College of Nuclear Technology & Chemistry and BiologyHubei University of Science and Technology Xianning China

4. Department of Nuclear Medicine and PET/CT-MRI Centerthe First Affiliated Hospital of Jinan University & Institute of Molecular and Functional ImagingJinan University Guangzhou 510630 China

5. Department of Chemistry and BiochemistryUniversity of Oklahoma Norman OK 73019 USA

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1002/cmdc.201800710

Reference46 articles.

1. Molecular Biology of Muscarinic Acetylcholine Receptors

2. Muscarinic acetylcholine receptor subtypes in cerebral cortex and hippocampus

3. Muscarinic Acetylcholine Receptors

4. Muscarinic receptors: their distribution and function in body systems, and the implications for treating overactive bladder

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