Selective Neutral pH Inhibitor of Cathepsin B Designed Based on Cleavage Preferences at Cytosolic and Lysosomal pH Conditions

Author:

Yoon Michael C.12ORCID,Solania Angelo3ORCID,Jiang Zhenze1ORCID,Christy Mitchell P.4,Podvin Sonia1,Mosier Charles1,Lietz Christopher B.1,Ito Gen1,Gerwick William H.4,Wolan Dennis W.3ORCID,Hook Gregory5,O’Donoghue Anthony J.1,Hook Vivian16ORCID

Affiliation:

1. Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California, San Diego, La Jolla, California 92093, United States

2. Biomedical Sciences Graduate Program, University of California, San Diego, La Jolla, California 92093, United States

3. Departments of Molecular Medicine and Integrative Structural and Computational Biology, The Scripps Research Institute, La Jolla, California 92037, United States

4. Scripps Institution of Oceanography, University of California, San Diego, La Jolla, California 92093, United States

5. American Life Sciences Pharmaceuticals, Inc., La Jolla, California 92037, United States

6. Department of Neurosciences, School of Medicine, University of California, San Diego, La Jolla, California 92037, United States

Funder

National Institute of Neurological Disorders and Stroke

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

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