Potent Inhibitors of Acetyltransferase Eis Overcome Kanamycin Resistance in Mycobacterium tuberculosis-Reference-Cited by-同舟云学术

Potent Inhibitors of Acetyltransferase Eis Overcome Kanamycin Resistance in Mycobacterium tuberculosis

Published:2016-04-07 Issue:6 Volume:11 Page:1639-1646
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Willby Melisa J.¹,Green Keith D.²,Gajadeera Chathurada S.²,Hou Caixia²,Tsodikov Oleg V.²,Posey James E.¹,Garneau-Tsodikova Sylvie²

Affiliation:

1. Division of Tuberculosis Elimination, National Center for HIV/AIDS, Viral Hepatitis, STD, and TB Prevention, Centers for Disease Control and Prevention, Atlanta, Georgia 30329, United States

2. Department of Pharmaceutical Sciences, University of Kentucky, Lexington, Kentucky 40536-0596, United States

Funder

National Institute of Allergy and Infectious Diseases

Firland Foundation

Argonne National Laboratory, Office of Science

College of Pharmacy, University of Kentucky

Center for Chemical Genomics, University of Michigan

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acschembio.6b00110

Reference35 articles.

1. World Health Organization (2014) Global Tuberculosis Report 2014. ISBM 978 992 974 156580 156589.

2. Resistance in tuberculosis: what do we know and where can we go?

3. Molecular Detection of Mutations Associated with First- and Second-Line Drug Resistance Compared with Conventional Drug Susceptibility Testing of Mycobacterium tuberculosis

4. Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB

5. Aminoglycoside Multiacetylating Activity of the Enhanced Intracellular Survival Protein from Mycobacterium smegmatis and Its Inhibition

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