Discovery and Mechanistic Analysis of Structurally Diverse Inhibitors of Acetyltransferase Eis among FDA-Approved Drugs
Author:
Affiliation:
1. Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, 789 South Limestone Street, Lexington, Kentucky40536-0596, United States
Funder
National Institute of Allergy and Infectious Diseases
Firland Foundation
College of Pharmacy, University of Kentucky
Center for Chemical Genomics, University of Michigan
Publisher
American Chemical Society (ACS)
Subject
Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.biochem.2c00658
Reference37 articles.
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2. Tuberculosis — United States, 2020
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5. Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
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