C–N Coupling of DNA-Conjugated (Hetero)aryl Bromides and Chlorides for DNA-Encoded Chemical Library Synthesis-Reference-Cited by-同舟云学术

C–N Coupling of DNA-Conjugated (Hetero)aryl Bromides and Chlorides for DNA-Encoded Chemical Library Synthesis

Published:2020-02-05 Issue:3 Volume:31 Page:770-780
ISSN:1043-1802
Container-title:Bioconjugate Chemistry
language:en
Short-container-title:Bioconjugate Chem.

Author:

Chen Ying-Chu¹,Faver John C.¹,Ku Angela F.¹,Miklossy Gabriella¹,Riehle Kevin¹,Bohren Kurt M.¹,Ucisik Melek N.¹,Matzuk Martin M.¹,Yu Zhifeng¹,Simmons Nicholas¹^ORCID

Affiliation:

1. Center for Drug Discovery, Department of Pathology and Immunology, Baylor College of Medicine, Houston, Texas 77030, United States

Funder

Welch Foundation

Bill and Melinda Gates Foundation

Eunice Kennedy Shriver National Institute of Child Health and Human Development

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Pharmaceutical Science,Pharmacology,Biomedical Engineering,Bioengineering,Biotechnology

Link

http://pubs.acs.org/doi/pdf/10.1021/acs.bioconjchem.9b00863

Reference54 articles.

1. DNA-encoded chemistry: enabling the deeper sampling of chemical space

2. DNA-Encoded Chemical Libraries: A Selection System Based on Endowing Organic Compounds with Amplifiable Information

3. Discovery of Small-Molecule Interleukin-2 Inhibitors from a DNA-Encoded Chemical Library

4. DNA-Encoded Library Screening Identifies Benzo[b][1,4]oxazepin-4-ones as Highly Potent and Monoselective Receptor Interacting Protein 1 Kinase Inhibitors

5. Discovery of a First-in-Class Receptor Interacting Protein 1 (RIP1) Kinase Specific Clinical Candidate (GSK2982772) for the Treatment of Inflammatory Diseases

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