DNA-Encoded Library Screening Identifies Benzo[b][1,4]oxazepin-4-ones as Highly Potent and Monoselective Receptor Interacting Protein 1 Kinase Inhibitors-Reference-Cited by-同舟云学术

DNA-Encoded Library Screening Identifies Benzo[b][1,4]oxazepin-4-ones as Highly Potent and Monoselective Receptor Interacting Protein 1 Kinase Inhibitors

Published:2016-02-23 Issue:5 Volume:59 Page:2163-2178
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Harris Philip A.,King Bryan W.,Bandyopadhyay Deepak,Berger Scott B.,Campobasso Nino,Capriotti Carol A.,Cox Julie A.,Dare Lauren,Dong Xiaoyang,Finger Joshua N.,Grady LaShadric C.¹,Hoffman Sandra J.,Jeong Jae U.,Kang James,Kasparcova Viera,Lakdawala Ami S.,Lehr Ruth,McNulty Dean E.,Nagilla Rakesh,Ouellette Michael T.,Pao Christina S.,Rendina Alan R.,Schaeffer Michelle C.,Summerfield Jennifer D.¹,Swift Barbara A.,Totoritis Rachel D.,Ward Paris,Zhang Aming²,Zhang Daohua,Marquis Robert W.,Bertin John,Gough Peter J.

Affiliation:

1. Platform Technology & Science, GlaxoSmithKline, Winter Street, Waltham, Massachusetts 02451, United States

2. Platform Technology & Science, GlaxoSmithKline, King of Prussia, Pennsylvania 19406, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5b01898

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