A Non-Peptide NK1 Receptor Agonist Showing Subpicomolar Affinity-Reference-Cited by-同舟云学术

A Non-Peptide NK1 Receptor Agonist Showing Subpicomolar Affinity

Published:2004-02-11 Issue:6 Volume:47 Page:1315-1318
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Cappelli Andrea¹,Giuliani Germano¹,Pericot Mohr Gal.la¹,Gallelli Andrea¹,Anzini Maurizio¹,Vomero Salvatore¹,Cupello Aroldo¹,Scarrone Simona¹,Matarrese Mario¹,Moresco Rosa Maria¹,Fazio Ferruccio¹,Finetti Federica¹,Morbidelli Lucia¹,Ziche Marina¹

Affiliation:

1. Dipartimento Farmaco Chimico Tecnologico and European Research Centre for Drug Discovery and Development, Università degli Studi di Siena, Via A. Moro, 53100 Siena, Italy, Istituto di Bioimmagini e Fisiologia Molecolare, CNR, Sezione di Genova, Via de Toni 5, 16132 Genova, Italy, Istituto di Bioimmagini e Fisiologia Molecolare, CNR, Istituto H. S. Raffaele, Università di Milano/Bicocca, Via Olgettina 60, 20132 Milano, Italy, and Sezione di Farmacologia, Dipartimento di Biologia Molecolare, Università...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm034219a

Reference16 articles.

1. Substance P: a pioneer amongst neuropeptides

2. A Potent Nonpeptide Antagonist of the Substance P (NK 1 ) Receptor

3. Novel, Potent, and Orally Active Substance P Antagonists: Synthesis and Antagonist Activity of N-Benzylcarboxamide Derivatives of Pyrido[3,4-b]pyridine

4. Nonpeptide Cholecystokinin-2 Receptor Agonists

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