Design, synthesis and biological studies of a library of NK1-Receptor Ligands Based on a 5-arylthiosubstituted 2-amino-4,6-diaryl-3-cyano-4 H -pyran core: Switch from antagonist to agonist effect by chemical modification-Reference-Cited by-同舟云学术

Design, synthesis and biological studies of a library of NK1-Receptor Ligands Based on a 5-arylthiosubstituted 2-amino-4,6-diaryl-3-cyano-4 H -pyran core: Switch from antagonist to agonist effect by chemical modification

Published:2017-09 Issue: Volume:138 Page:644-660
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Recio Rocío,Vengut-Climent Empar,Mouillac Bernard,Orcel Hélène,López-Lázaro Miguel,Calderón-Montaño José Manuel,Álvarez Eleuterio,Khiar Noureddine,Fernández Inmaculada

Funder

Spanish Ministerio de Economía y Competitividad (MEC)

Junta de Andalucía

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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