Bioisosteric Modifications of 2-Arylureidobenzoic Acids: Selective Noncompetitive Antagonists for the Homomeric Kainate Receptor Subtype GluR5-Reference-Cited by-同舟云学术

Bioisosteric Modifications of 2-Arylureidobenzoic Acids: Selective Noncompetitive Antagonists for the Homomeric Kainate Receptor Subtype GluR5

Published:2004-12-01 Issue:27 Volume:47 Page:6948-6957
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Valgeirsson Jon¹,Nielsen Elsebet Ø.¹,Peters Dan¹,Mathiesen Claus¹,Kristensen Anders S.¹,Madsen Ulf¹

Affiliation:

1. Department of Medicinal Chemistry and Department of Pharmacology, The Danish University of Pharmaceutical Sciences, 2 Universitetsparken, DK-2100 Copenhagen, Denmark, and NeuroSearch A/S, 93 Pederstrupvej, DK-2750 Ballerup, Denmark

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030638w

Reference34 articles.

1. Ligands for Glutamate Receptors: Design and Therapeutic Prospects

2. Glutamate in CNS disorders as a target for drug development: an update

3. Decahydroisoquinolines: novel competitive AMPA/kainate antagonists with neuroprotective effects in global cerebral ischaemia

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