Quinoxalinylethylpyridylthioureas (QXPTs) as Potent Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further SAR Studies and Identification of a Novel Orally Bioavailable Hydrazine-Based Antiviral Agent-Reference-Cited by-同舟云学术

Quinoxalinylethylpyridylthioureas (QXPTs) as Potent Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further SAR Studies and Identification of a Novel Orally Bioavailable Hydrazine-Based Antiviral Agent

Published:2001-01-03 Issue:3 Volume:44 Page:305-315
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Campiani Giuseppe¹,Aiello Francesca¹,Fabbrini Monica¹,Morelli Elena¹,Ramunno Anna¹,Armaroli Silvia¹,Nacci Vito¹,Garofalo Antonio¹,Greco Giovanni¹,Novellino Ettore¹,Maga Giovanni¹,Spadari Silvio¹,Bergamini Alberto¹,Ventura Laura¹,Bongiovanni Barbara¹,Capozzi Marcella¹,Bolacchi Francesca¹,Marini Stefano¹,Coletta Massimiliano¹,Guiso Giovanna¹,Caccia Silvio¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche, Facolta' di Farmacia, Universita' degli Studi di Salerno, via Ponte Don Melillo 11C, 84084 Fisciano (Salerno), Italy, Dipartimento Farmaco Chimico Tecnologico, Universita' degli Studi di Siena, via Aldo Moro, 53100 Siena, Italy, Universita' della Calabria, 87036 Arcavacata, Cosenza, Italy, Dipartimento di Chimica Farmaceutica e Tossicologica, Universita' di Napoli “Federico II”, via D. Montesano 49, 80131 Napoli, Italy, Istituto di Genetica Biochimica ed...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0010365

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1. Isolation of a T-Lymphotropic Retrovirus from a Patient at Risk for Acquired Immune Deficiency Syndrome (AIDS)

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3. Antiviral Therapy in Human Immunodeficiency Virus Infections

4. Potent and selective inhibition of HIV-1 replication in vitro by a novel series of TIBO derivatives

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