Copper-catalyzed oxidative cyclization of 2-(1<i>H</i>-pyrrol-1-yl)aniline and alkylsilyl peroxides: a route to pyrrolo[1,2-<i>a</i>]quinoxalines-Reference-Cited by-同舟云学术

Copper-catalyzed oxidative cyclization of 2-(1H-pyrrol-1-yl)aniline and alkylsilyl peroxides: a route to pyrrolo[1,2-a]quinoxalines

Published:2024 Issue:12 Volume:22 Page:2370-2374
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

An Zhenyu¹^ORCID,Miao Man¹,Sun Fengkai¹,Lan Xiao-Bing¹,Yu Jian-Qiang¹^ORCID,Guo Xiaoli¹,Zhang Jian¹²^ORCID

Affiliation:

1. College of Pharmacy, Key Laboratory of Protection, Development and Utilization of Medicinal Resources in Liupanshan Area, Ministry of Education, Ningxia Medical University, Yinchuan, Ningxia Hui Autonomous Region, China

2. Medicinal Chemistry and Bioinformatics Center, Shanghai Jiao Tong University School of Medicine, Shanghai, China

Abstract

An efficient method was developed for the one-pot construction of pyrrolo[1,2-a]quinoxalines via a Cu(ii)-catalyzed domino reaction between 2-(1H-pyrrol-1-yl)anilines and alkylsilyl peroxides.

Funder

Natural Science Foundation of Ningxia Province

Ningxia Medical University

National Basic Research Program of China

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/OB/D3OB01934A

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