Eleven Amino Acid Glucagon-like Peptide-1 Receptor Agonists with Antidiabetic Activity

Author:

Mapelli Claudio1,Natarajan Sesha I.1,Meyer Jean-Philippe1,Bastos Margarita M.1,Bernatowicz Michael S.1,Lee Ving G.1,Pluscec Jelka1,Riexinger Douglas J.1,Sieber-McMaster Ellen S.1,Constantine Keith L.1,Smith-Monroy Constance A.2,Golla Rajasree2,Ma Zhengping2,Longhi Daniel A.2,Shi Dan3,Xin Li2,Taylor Joseph R.2,Koplowitz Barry4,Chi Cecilia L.4,Khanna Ashish4,Robinson Gordon W.2,Seethala Ramakrishna2,Antal-Zimanyi Ildiko A.2,Stoffel Robert H.3,Han Songping2,Whaley Jean M.2,Huang Christine S.4,Krupinski John2,Ewing William R.5

Affiliation:

1. Department of Applied Biotechnologies, Bristol-Myers Squibb Company Research & Development, Princeton, New Jersey 08543

2. Diabetes Drug Discovery

3. Department of Applied Biotechnologies

4. Preclinical Candidate Optimization

5. Discovery Chemistry

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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