Enantiopure Cyclopropane-Bearing Pyridyldiazabicyclo[3.3.0]octanes as Selective α4β2-nAChR Ligands-Reference-Cited by-同舟云学术

Enantiopure Cyclopropane-Bearing Pyridyldiazabicyclo[3.3.0]octanes as Selective α4β2-nAChR Ligands

Published:2014-10-01 Issue:11 Volume:5 Page:1196-1201
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Onajole Oluseye K.¹,Eaton J. Brek²,Lukas Ronald J.²,Brunner Dani³,Thiede Lucinda³,Caldarone Barbara J.⁴,Kozikowski Alan P.¹

Affiliation:

1. Department of Medicinal Chemistry and Pharmacognosy, College of Pharmacy, University of Illinois at Chicago, 833 South Wood Street, Chicago, Illinois 60612, United States

2. Division of Neurobiology, Barrow Neurological Institute, 350 West Thomas Road, Phoenix, Arizona 85013, United States

3. PsychoGenics, Inc., 765 Old Saw Mill River Road, Tarrytown, New York 10591, United States

4. NeuroBehavior Laboratory, Harvard NeuroDiscovery Center and Department of Neurology, Brigham and Women’s Hospital, 77 Avenue Louis Pasteur, Boston, Massachusetts 02115, United States

Funder

National Institute of Mental Health

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml500129k

Reference31 articles.

1. Structural and functional diversity of native brain neuronal nicotinic receptors

2. Brain Neuronal Nicotinic Receptors as New Targets for Drug Discovery

3. Central Nicotinic Receptors: Structure, Function, Ligands, and Therapeutic Potential