Design, Synthesis, and Pharmacological Evaluation of a Novel Series of Pyridopyrazine-1,6-dione γ-Secretase Modulators-Reference-Cited by-同舟云学术

Design, Synthesis, and Pharmacological Evaluation of a Novel Series of Pyridopyrazine-1,6-dione γ-Secretase Modulators

Published:2014-01-28 Issue:3 Volume:57 Page:1046-1062
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Pettersson Martin¹,Johnson Douglas S.¹,Subramanyam Chakrapani²,Bales Kelly R.¹,am Ende Christopher W.²,Fish Benjamin A.²,Green Michael E.¹,Kauffman Gregory W.¹,Mullins Patrick B.²,Navaratnam Thayalan²,Sakya Subas M.²,Stiff Cory M.²,Tran Tuan P.²,Xie Longfei²,Zhang Liming²,Pustilnik Leslie R.²,Vetelino Beth C.²,Wood Kathleen M.¹,Pozdnyakov Nikolay¹,Verhoest Patrick R.¹,O’Donnell Christopher J.²

Affiliation:

1. Pfizer Worldwide Research & Development, 610 Main Street, Cambridge, Massachusetts 02139, United States

2. Pfizer Worldwide Research & Development, Eastern Point Road, Groton, Connecticut 06340, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm401782h

Reference62 articles.

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