Structural Characterization of Thiadiazolesulfonamide Inhibitors Bound to <i>Neisseria gonorrhoeae</i> α-Carbonic Anhydrase-Reference-Cited by-同舟云学术

Structural Characterization of Thiadiazolesulfonamide Inhibitors Bound to Neisseria gonorrhoeae α-Carbonic Anhydrase

Published:2022-12-06 Issue:1 Volume:14 Page:103-109
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Marapaka Anil Kumar¹^ORCID,Nocentini Alessio²^ORCID,Youse Molly S.¹,An Weiwei¹,Holly Katrina J.¹,Das Chittaranjan³^ORCID,Yadav Ravi⁴,Seleem Mohamed N.⁵^ORCID,Supuran Claudiu T.²^ORCID,Flaherty Daniel P.¹^ORCID

Affiliation:

1. Department of Medicinal Chemistry and Molecular Pharmacology, College of Pharmacy, Purdue University, West Lafayette, Indiana47907, United States

2. Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Polo Scientifico, Firenze50122, Italy

3. Department of Chemistry, College of Sciences, Purdue University, West Lafayette, Indiana47907, United States

4. Department of Biological Sciences, College of Sciences, Purdue University, West Lafayette, Indiana47907, United States

5. Department of Biomedical Sciences and Pathobiology, Virginia-Maryland College of Veterinary Medicine, Virginia Polytechnic Institute and State University, Blacksburg, Virginia24061, United States

Funder

Ministero dell?Istruzione, dell?Universit? e della Ricerca

National Institute of Allergy and Infectious Diseases

Purdue Institute for Drug Discovery

Purdue College of Pharmacy

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.2c00471

Reference31 articles.

1. Multi-drug resistant gonorrhoeae fact sheet. World Health Organization, Geneva, Switzerland, Aug 25, 2020. https://www.who.int/news-room/fact-sheets/detail/multi-drug-resistant-gonorrhoea.

2. Sexually Transmitted Disease Surveillance 2020. Centers for Disease Control and Prevention, Atlanta, GA, 2020. https://www.cdc.gov/std/statistics/2020/overview.htm#Gonorrhea (page last reviewed: April 12, 2022).

3. Antibiotic Resistance Threats in the United States, 2019; Centers for Disease Control and Prevention, Atlanta, GA, December 2019. https://www.cdc.gov/drugresistance/pdf/threats-report/2019-ar-threats-report-508.pdf.

4. Antimicrobial resistance in Neisseria gonorrhoeae: Global surveillance and a call for international collaborative action

5. Update to CDC's Treatment Guidelines for Gonococcal Infection, 2020

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