Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae

Author:

Bonardi Alessandro1,Nocentini Alessio1ORCID,Giovannuzzi Simone1,Paoletti Niccolò1ORCID,Ammara Andrea1ORCID,Bua Silvia2,Abutaleb Nader S.3,Abdelsattar Abdallah S.3,Capasso Clemente4,Gratteri Paola1ORCID,Flaherty Daniel P.5ORCID,Seleem Mohamed N.36ORCID,Supuran Claudiu T.1ORCID

Affiliation:

1. NEUROFARBA Department, Pharmaceutical and Nutraceutical Section and Laboratory of Molecular Modeling Cheminformatics & QSAR, University of Florence, Via U. Schiff 6, Sesto Fiorentino, Florence 50019, Italy

2. Research Institute of the University of Bucharest (ICUB), Bucharest 050663, Romania

3. Department of Biomedical Sciences and Pathobiology, Virginia-Maryland College of Veterinary Medicine, Virginia Polytechnic Institute and State University, Blacksburg, Virginia 24061, United States

4. Istituto di Bioscienze e Biorisorse, CNR, Naples 80131, Italy

5. Borch Department of Medicinal Chemistry and Molecular Pharmacology, College of Pharmacy, Purdue University, West Lafayette, Indiana 47907, United States

6. Center for One Health Research, Virginia Polytechnic Institute and State University, Blacksburg, Virginia 24061, United States

Funder

Research Institute, University of Bucharest

European Commission

National Institute of Allergy and Infectious Diseases of the National Institutes of Health

NextGenerationEU

Publisher

American Chemical Society (ACS)

Cited by 3 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献

1. Fighting antibacterial drug resistance;Expert Opinion on Therapeutic Patents;2024-06-02

2. Management of Neisseria gonorrhoeae infection: from drug resistance to drug repurposing;Expert Opinion on Therapeutic Patents;2024-06-02

3. Sulfonamide inhibitors of bacterial carbonic anhydrases;The Enzymes;2024

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