From PARP1 to TNKS2 Inhibition: A Structure-Based Approach-Reference-Cited by-同舟云学术

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From PARP1 to TNKS2 Inhibition: A Structure-Based Approach

Published:2020-02-03 Issue:5 Volume:11 Page:862-868
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Tomassi Stefano¹^ORCID,Pfahler Julian²,Mautone Nicola³,Rovere Annarita³,Esposito Chiara⁴,Passeri Daniela⁵,Pellicciari Roberto⁵,Novellino Ettore¹^ORCID,Pannek Martin²,Steegborn Clemens²^ORCID,Paiardini Alessandro⁴,Mai Antonello³^ORCID,Rotili Dante³

Affiliation:

1. Department of Pharmacy, University of Naples, “Federico II”, 80131 Naples, Italy

2. Department of Biochemistry and Research Center for Bio-Macromolecules, University of Bayreuth, 95440 Bayreuth, Germany

3. Department of Chemistry and Technology of Drugs, ″Sapienza” University of Rome, 00185 Rome, Italy

4. Department of Biochemical Sciences “A. Rossi Fanelli″, ″Sapienza” University of Rome, 00185 Rome, Italy

5. TES Pharma S.r.l., 06073 Corciano, Perugia, Italy

Funder

Ministero dell?Istruzione, dell?Universit? e della Ricerca

Associazione Italiana per la Ricerca sul Cancro

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.9b00654

Reference22 articles.

1. Toward a unified nomenclature for mammalian ADP-ribosyltransferases

2. PARP family enzymes: regulation and catalysis of the poly(ADP-ribose) posttranslational modification

3. Tankyrase-targeted therapeutics: expanding opportunities in the PARP family

4. Regulation of Wnt/β-catenin signalling by tankyrase-dependent poly(ADP-ribosyl)ation and scaffolding

5. Novel insight into the function of tankyrase (Review)

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1. Discovering Dually Active Anti-cancer Compounds with a Hybrid AI-structure-based Approach;Journal of Chemical Information and Modeling;2024-09-14

2. Probing intracellular determinants of PARP inhibitor selectivity and pharmacology with CeTEAM;2024-08-10

3. Chain Extension of Piperazine in Ethanol: Synthesis of 2-(4-(2-(Phenylthio)ethyl)piperazinyl)acetonitriles and ACAT-1 Inhibitors;Molecules;2024-08-06

4. Blue LED Induced Three Component Reactions for the Generation of 4,6‐Dioxo‐hexahydro‐1H‐furo[3, 4‐c] pyrrole: Their Evaluation as Anticancer Agents through PARP‐1 Inhibition;Chemistry – An Asian Journal;2023-06-21

5. Selective PARP1 inhibitors, PARP1-based dual-target inhibitors, PROTAC PARP1 degraders, and prodrugs of PARP1 inhibitors for cancer therapy;Pharmacological Research;2022-12

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